URI:
   DIR Return Create A Forum - Home
       ---------------------------------------------------------
       MS Speaks
  HTML https://msspeaks.createaforum.com
       ---------------------------------------------------------
       *****************************************************
   DIR Return to: AUBAGIO (teriflunomide)
       *****************************************************
       #Post#: 457--------------------------------------------------
       Aubagio for patients w/1st clinical episode suggesting MS: TOPIC
       phase 3 study
   DIR By: agate
       Date: September 5, 2014, 7:28 pm
       ---------------------------------------------------------
       From Science Direct (September 3) citing The Lancet Neurology,
       September 2, 2014:
       --- Quote ---
       >
       >
       > The Lancet Neurology
       > Available online 2 September 2014
       > In Press, Corrected Proof
       >
       > Oral teriflunomide for patients with a first clinical episode
       suggestive of multiple sclerosis (TOPIC): a randomised,
       double-blind, placebo-controlled, phase 3 trial
       >
       > Prof Aaron E Miller, MD,  Prof Jerry S Wolinsky, MD, Ludwig
       Kappos, MD, Prof Giancarlo Comi, MD, Prof Mark S Freedman, MDe,
       Prof Tomas P Olsson, MDf, Deborah Bauer, MS, Myriam Benamor, MD,
       Philippe Truffinet, MD, Prof Paul W O'Connor, MD, for the TOPIC
       Study Group
       >
       > Summary
       >
       > Background
       >
       > Teriflunomide is a once-daily oral immunomodulator approved
       for the treatment of relapsing-remitting multiple sclerosis. We
       aimed to assess the efficacy and safety of teriflunomide in
       patients with a first clinical episode suggestive of multiple
       sclerosis.
       >
       > Methods
       >
       > In this randomised, double-blind, placebo-controlled,
       parallel-group study, we enrolled patients aged 18–55 years with
       clinically isolated syndrome (defined as a neurological event
       consistent with demyelination, starting within 90 days of
       randomisation, and two or more T2-weighted MRI lesions ≥3
       mm in diameter) from 112 centres (mostly hospitals) in 20
       countries. Participants were randomly assigned (1:1:1) in a
       double-blind manner (by an interactive voice response system) to
       once-daily oral teriflunomide 14 mg, teriflunomide 7 mg, or
       placebo, for up to 108 weeks. Patients, staff administering the
       interventions, and outcome assessors were masked to treatment
       assignment.
       >
       > The primary endpoint was time to relapse (a new neurological
       abnormality separated by ≥30 days from a preceding
       clinical event, present for ≥24 h in the absence of fever
       or known infection), which defined conversion to clinically
       definite multiple sclerosis.
       >
       > The key secondary endpoint was time to relapse or new
       gadolinium-enhancing or T2 lesions on MRI, whichever occurred
       first.
       >
       > The primary outcome was analysed for the modified
       intention-to-treat population; safety analyses included all
       randomised patients who were exposed to the study drug, as
       treated.
       >
       > This trial is registered with ClinicalTrials.gov, number
       NCT00622700.
       >
       > Findings
       >
       > Between Feb 13, 2008, and Aug 22, 2012, 618 patients were
       enrolled and randomly assigned to teriflunomide 14 mg (n=216),
       teriflunomide 7 mg (n=205), or placebo (n=197). Two patients in
       each of the teriflunomide groups did not receive the study drug,
       so the modified intention-to-treat population comprised 214
       patients in the teriflunomide 14 mg group, 203 in the
       teriflunomide 7 mg group, and 197 in the placebo group. Compared
       with placebo, teriflunomide significantly reduced the risk of
       relapse defining clinically definite multiple sclerosis at the
       14 mg dose (hazard ratio [HR] 0·574 [95% CI 0·379–0·869];
       p=0·0087) and at the 7 mg dose (0·628 [0·416–0·949]; p=0·0271).
       Teriflunomide reduced the risk of relapse or a new MRI lesion
       compared with placebo at the 14 mg dose (HR 0·651 [95% CI
       0·515–0·822]; p=0·0003) and at the 7 mg dose (0·686
       [0·540–0·871]; p=0·0020). During the study, six patients who
       were randomly assigned to placebo accidently also received
       teriflunomide at some point: four received 7 mg and two received
       14 mg. Therefore, the safety population comprised 216 patients
       on teriflunomide 14 mg, 207 on teriflunomide 7 mg, and 191 on
       placebo.
       >
       > Adverse events that occurred in at least 10% of patients in
       either teriflunomide group and with an incidence that was at
       least 2% higher than that with placebo were increased alanine
       aminotransferase (40 [19%] of 216 patients in the 14 mg group,
       36 [17%] of 207 in the 7 mg group vs 27 [14%] of 191 in the
       placebo group), hair thinning (25 [12%] and 12 [6%] vs 15 [8%]),
       diarrhoea (23 [11%] and 28 [14%] vs 12 [6%]), paraesthesia (22
       [10%] and 11 [5%] vs 10 [5%]), and upper respiratory tract
       infection (20 [9%] and 23 [11%] vs 14 [7%]). The most common
       serious adverse event was an increase in alanine
       aminotransferase (four [2%] and five [2%] vs three [2%]).
       >
       > Interpretation
       >
       > TOPIC is to our knowledge the first study to report benefits
       of an available oral disease-modifying therapy in patients with
       early multiple sclerosis. These results extend the stages of
       multiple sclerosis in which teriflunomide shows a beneficial
       effect.
       >
       > Funding
       >
       > Genzyme, a Sanofi company.
       >
       > Correspondence to:
       >
       > Prof Aaron E Miller, Icahn School of Medicine at Mount Sinai,
       The Corinne Goldsmith Dickinson Center for Multiple Sclerosis, 5
       East 98th Street; Box 1138, New York, NY 10029, USA
       >
       --- End Quote ---
       The article is available here
  HTML http://www.sciencedirect.com/science/article/pii/S1474442214701917.
       *****************************************************
       Page 1 of 1